SCHEMBL13862003

SCHEMBL13862003

CC(CO)c1ccc(C(=O)Nc2cn3cc(Cl)ccc3n2)cc1

nearest known ligand 0.67

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 15/20 0.67
RET P07949 2/20 0.43
CDK2 P24941 2/20 0.43
GSK3B P49841 2/20 0.43
ITK Q08881 2/20 0.43
MERTK Q12866 2/20 0.43
PRKAA1 Q13131 2/20 0.43
ROCK1 Q13464 2/20 0.43
MAP3K6 O95382 2/20 0.42
CYP2C19 P33261 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
KDM4E B2RXH2 1/20 0.41
TP53 P04637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3486443 0.81 MAP3K5 (0.79) MAP3K5RETCDK2GSK3BITK
SCHEMBL3486097 0.80 MAP3K5 (1.00) MAP3K5RETCDK2GSK3BITK
Hydrochloric Acid SCHEMBL3486202 0.80 MAP3K5 (0.77) MAP3K5RETCDK2GSK3BITK
SCHEMBL3486350 0.79 MAP3K5 (0.84) MAP3K5RETCDK2GSK3BITK
SCHEMBL3486275 0.79 MAP3K5 (0.76) MAP3K5RETCDK2GSK3BITK
SCHEMBL3485910 0.78 MAP3K5 (0.77) MAP3K5RETCDK2GSK3BITK
SCHEMBL3486220 0.77 MAP3K5 (0.80) MAP3K5RETCDK2GSK3BITK
SCHEMBL3485624 0.77 MAP3K5 (0.65) MAP3K5RETCDK2GSK3BITK
SCHEMBL3486197 0.77 MAP3K5 (0.65) MAP3K5RETCDK2GSK3BITK
SCHEMBL3486068 0.77 MAP3K5 (0.65) MAP3K5CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2058309-A1 FUSED HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2009-05-13 EP disclosed