SCHEMBL13865175

SCHEMBL13865175

CCOC(=O)c1coc(-c2nn(Cc3ccccc3)c3ccccc23)n1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2RL3 Q96RI0 1/20 0.63
CYP2D6 P10635 7/20 0.48
CYP1A2 P05177 5/20 0.48
PDE5A O76074 4/20 0.48
CYP3A4 P08684 2/20 0.48
SCN8A Q9UQD0 1/20 0.48
ALDH1A1 P00352 3/20 0.45
MAPK1 P28482 2/20 0.45
SMN1; SMN2 Q16637 3/20 0.44
LMNA P02545 2/20 0.44
CYP19A1 P11511 2/20 0.44
KDM4E B2RXH2 1/20 0.44
NPC1 O15118 1/20 0.44
GMNN O75496 1/20 0.44
TP53 P04637 1/20 0.44
MAPT P10636 1/20 0.44
CYP2C9 P11712 1/20 0.44
HPGD P15428 1/20 0.44
ALOX15 P16050 1/20 0.44
NFKB1 P19838 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5430238 0.80 F2RL3 (0.64) F2RL3CYP2D6CYP1A2PDE5ACYP3A4
SCHEMBL7660191 0.80 F2RL3 (0.63) F2RL3CYP2D6CYP1A2PDE5ACYP3A4
SCHEMBL13865174 0.78 CYP2D6 (0.56) F2RL3CYP2D6CYP1A2PDE5ACYP3A4
SCHEMBL3245414 0.78 F2RL3 (0.67) F2RL3CYP2D6CYP1A2PDE5ACYP3A4
SCHEMBL363569 0.78 F2RL3 (1.00) F2RL3PDE5AALDH1A1MAPK1SMN1; SMN2
SCHEMBL29403731 0.78 F2RL3 (1.00) F2RL3PDE5AALDH1A1MAPK1SMN1; SMN2
SCHEMBL18427929 0.78 F2RL3 (0.69) F2RL3CYP2D6CYP1A2PDE5ACYP3A4
SCHEMBL5558869 0.76 CYP2D6 (0.57) F2RL3CYP2D6CYP1A2PDE5ACYP3A4
SCHEMBL7488323 0.75 F2RL3 (0.78) F2RL3PDE5AALDH1A1SMN1; SMN2LMNA
SCHEMBL13865197 0.75 CYP2D6 (0.55) F2RL3CYP2D6CYP1A2PDE5ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934311-B1 NEW HETEROCYCLYLMETHYL-SUBSTITUTED PYRAZOL DERIVATES BAYER HEALTHCARE AG (DE) 2009-05-13 EP disclosed