SCHEMBL1387488

SCHEMBL1387488

COc1nc(Br)cnc1NS(=O)(=O)c1cc(C)ccc1-c1ccccc1

nearest known ligand 0.78

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 7/20 0.78
CCR4 P51679 13/20 0.64
CCR5 P51681 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1387415 0.88 EDNRA (1.00) EDNRACCR4CCR5
SCHEMBL7948489 0.87 EDNRA (0.85) EDNRACCR4CCR5
SCHEMBL1387374 0.81 EDNRA (0.85) EDNRACCR4CCR5
SCHEMBL1731921 0.78 CCR4 (1.00) EDNRACCR4CCR5
SCHEMBL6038631 0.78 CCR4 (0.58) EDNRACCR4
SCHEMBL1387150 0.78 EDNRA (0.77) EDNRACCR4
SCHEMBL1731970 0.77 CCR4 (0.74) EDNRACCR4CCR5
SCHEMBL6039032 0.76 CCR4 (0.51) EDNRACCR4
SCHEMBL1387397 0.76 EDNRA (0.67) EDNRACCR4
SCHEMBL1387409 0.76 EDNRA (1.00) EDNRACCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-H09510987-A 1997-11-04 JP claimed
EP-0752986-A1 N-HETEROCYCLYL SULPHONAMIDE DERIVATIVES AND THEIR USE AS ENDOTHELIN ANTAGONISTS ZENECA LIMITED (GB) 1997-01-15 EP claimed
WO-1995026957-A1 N-HETEROCYCLYL SULPHONAMIDE DERIVATIVES AND THEIR USE AS ENDOTHELIN ANTAGONISTS ZENECA LIMITED (GB) 1995-10-12 WO claimed