SCHEMBL13893968

SCHEMBL13893968

Cc1ccc2c(=O)n(-c3cccc(-c4cc(Nc5ccc(C(=O)N6CCOCC6)cn5)c(=O)n(C)n4)c3C)cnc2c1

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BTK Q06187 17/20 0.60
KDM4E B2RXH2 1/20 0.49
RAB9A P51151 1/20 0.49
CLK2 P49760 1/20 0.45
TYK2 P29597 1/20 0.44
HPGD P15428 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8737222 0.93 BTK (0.58) BTKKDM4ERAB9ACLK2TYK2
SCHEMBL106616 0.92 BTK (0.66) BTKCLK2
SCHEMBL3804473 0.82 BTK (0.63) BTKKDM4ERAB9ACLK2TYK2
SCHEMBL3660016 0.81 BTK (0.62) BTKKDM4ERAB9ACLK2TYK2
SCHEMBL710063 0.80 BTK (0.75) BTKKDM4ERAB9ACLK2
SCHEMBL16417074 0.79 BTK (0.57) BTKKDM4ERAB9ACLK2TYK2
SCHEMBL19594126 0.77 BTK (0.85) BTKCLK2
SCHEMBL104439 0.77 BTK (0.77) BTKCLK2
SCHEMBL2492566 0.77 BTK (0.60) BTKKDM4ERAB9ACLK2TYK2
SCHEMBL19593975 0.77 BTK (0.69) BTKKDM4ERAB9ACLK2TYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009053269-A1 NOVEL KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2009-04-30 WO disclosed