SCHEMBL13907682

SCHEMBL13907682

Cc1cc2cc(C(=O)NCC(=O)N3CCC(N4CCc5ccccc5NC4=O)CC3)ccc2[nH]1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
OXTR P30559 1/20 0.46
CALCRL Q16602 13/20 0.43
RAMP1 O60894 2/20 0.43
P2RY12 Q9H244 1/20 0.42
CYP3A4 P08684 2/20 0.41
HSD11B1 P28845 2/20 0.41
ALDH1A1 P00352 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13907943 0.84 CALCRL (0.47) CALCRLRAMP1CYP3A4HSD11B1ALDH1A1
SCHEMBL13907858 0.83 CALCRL (0.52) CALCRLRAMP1CYP3A4
SCHEMBL13907849 0.82 SMYD3 (0.48) CALCRLRAMP1CYP3A4
SCHEMBL13907847 0.82 CALCRL (0.47) CALCRLRAMP1CYP3A4
SCHEMBL13907848 0.82 CALCRL (0.45) CALCRLRAMP1CYP3A4
SCHEMBL13907843 0.82 CALCRL (0.43) CALCRLRAMP1CYP3A4
SCHEMBL13907685 0.82 CALCRL (0.41) CALCRLRAMP1CYP3A4HTTSMN1; SMN2
SCHEMBL13907973 0.81 CALCRL (0.43) CALCRLRAMP1CYP3A4
SCHEMBL13907684 0.81 CALCRL (0.46) CALCRLRAMP1CYP3A4HTTSMN1; SMN2
SCHEMBL13907687 0.81 POLB (0.47) CALCRLRAMP1CYP3A4ALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009034029-A2 1-SUBSTITUTED 4-HETEROCYCLYLPIPERIDINES FOR USE AS CGRP ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-03-19 WO disclosed