SCHEMBL13907908

SCHEMBL13907908

CC(C)NCc1cc(C(=O)O)cc(Br)c1N

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 1/20 0.40
GSK3B P49841 1/20 0.39
THRA P10827 2/20 0.36
THRB P10828 2/20 0.36
TPMT P51580 1/20 0.36
MEP1B Q16820 4/20 0.35
ALDH1A1 P00352 2/20 0.34
CCR5 P51681 1/20 0.34
ADRB2 P07550 2/20 0.33
LMNA P02545 2/20 0.33
GBA1 P04062 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CNR1 P21554 1/20 0.33
TBXA2R P21731 1/20 0.33
HRH2 P25021 1/20 0.33
SLC6A4 P31645 1/20 0.33
KCNH2 Q12809 1/20 0.33
HIF1A Q16665 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13907669 0.88 GSK3B (0.39) GSK3BALDH1A1CCR5ADRB2LMNA
SCHEMBL11179265 0.80 ESR1 (0.39) GSK3BALDH1A1ADRB2KMT2A
SCHEMBL11621429 0.79 TTR (0.40) TTRGSK3BTPMTALDH1A1ADRB2
Hydrochloric Acid SCHEMBL11624379 0.79 TTR (0.40) TTRGSK3BTHRATHRBTPMT
SCHEMBL13907703 0.78 GAA (0.45) ALDH1A1CCR5ADRB2LMNAGBA1
SCHEMBL11156879 0.78 ESR1 (0.42) ALDH1A1ADRB2LMNACYP1A2RAB9A
SCHEMBL11163314 0.77 ESR1 (0.41) ALDH1A1ADRB2LMNACYP1A2RAB9A
SCHEMBL11154050 0.77 ESR1 (0.41) ALDH1A1ADRB2LMNACYP1A2CYP2D6
SCHEMBL11164947 0.76 ESR1 (0.41) ALDH1A1ADRB2LMNACYP1A2CYP2D6
SCHEMBL27817855 0.74 TTR (0.47) TTRGSK3BTHRATHRBTPMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009034029-A2 1-SUBSTITUTED 4-HETEROCYCLYLPIPERIDINES FOR USE AS CGRP ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-03-19 WO disclosed