SCHEMBL13932995

SCHEMBL13932995

COC(=O)c1ccc(OCCCc2ccc(OCCOc3ccccc3)cc2)c(C(=O)NC2CCCC(C(=O)OC)C2)c1

nearest known ligand 0.75

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYSLTR2 Q9NS75 2/20 0.75
RAB9A P51151 4/20 0.43
MAPT P10636 1/20 0.43
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
LTA4H P09960 3/20 0.39
POLB P06746 1/20 0.38
NPC1 O15118 2/20 0.38
OPRK1 P41145 1/20 0.38
FKBP1A P62942 1/20 0.37
SLC2A1 P11166 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4521894 0.98 CYSLTR2 (0.78) CYSLTR2RAB9AMAPTMEN1KMT2A
SCHEMBL4524350 0.96 CYSLTR2 (0.74) CYSLTR2RAB9AMAPTMEN1KMT2A
SCHEMBL4521604 0.94 CYSLTR2 (0.68) CYSLTR2RAB9AMAPTMEN1KMT2A
SCHEMBL4518460 0.94 CYSLTR2 (0.69) CYSLTR2RAB9AMAPTMEN1KMT2A
SCHEMBL13918309 0.94 CYSLTR2 (0.68) CYSLTR2MAPTMEN1KMT2AALDH1A1
SCHEMBL13918341 0.94 CYSLTR2 (0.70) CYSLTR2RAB9AMAPTMEN1KMT2A
SCHEMBL13918330 0.93 CYSLTR2 (0.68) CYSLTR2RAB9AMEN1KMT2AALDH1A1
SCHEMBL4520534 0.93 CYSLTR2 (0.68) CYSLTR2MAPTMEN1KMT2AALDH1A1
SCHEMBL13918239 0.92 CYSLTR2 (0.73) CYSLTR2RAB9AMAPTMEN1KMT2A
SCHEMBL4522056 0.92 CYSLTR2 (0.65) CYSLTR2RAB9AMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7498460-B2 Isophthalic acid derivatives BAYER HEALTHCARE AG (DE) 2009-03-03 US disclosed
EP-1572628-B1 ISOPHTALIC ACID DERIVATIVES BAYER HEALTHCARE AG (DE) 2007-07-25 EP disclosed