SCHEMBL13936619

SCHEMBL13936619

COc1cc2nccc(Oc3ccc(N(C)c4ccc(C(C)(C)C)cc4)cc3)c2cc1OC

nearest known ligand 0.82

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
FGFR2 P21802 14/20 0.82
PDGFRB P09619 2/20 0.60
PDGFRA P16234 2/20 0.60
KIT P10721 1/20 0.57
KDR P35968 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4484850 0.90 FGFR2 (1.00) FGFR2PDGFRBPDGFRAKITKDR
SCHEMBL5826095 0.86 FGFR2 (0.74) FGFR2PDGFRBPDGFRAKITKDR
SCHEMBL7489910 0.85 FGFR2 (0.76) FGFR2PDGFRBPDGFRAKITKDR
SCHEMBL8553216 0.85 FGFR2 (0.72) FGFR2PDGFRBPDGFRAKITKDR
SCHEMBL4473682 0.85 FGFR2 (0.84) FGFR2PDGFRBPDGFRAKITKDR
SCHEMBL4472020 0.85 FGFR2 (1.00) FGFR2PDGFRBPDGFRAKITKDR
SCHEMBL842293 0.83 FGFR2 (1.00) FGFR2PDGFRBPDGFRAKITKDR
SCHEMBL29574069 0.83 FGFR2 (1.00) FGFR2PDGFRBPDGFRAKITKDR
SCHEMBL4476013 0.83 FGFR2 (0.80) FGFR2PDGFRBPDGFRAKITKDR
SCHEMBL4473353 0.83 FGFR2 (0.80) FGFR2PDGFRBPDGFRAKITKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7495104-B2 Quinoline or quinazoline derivatives inhibiting auto-phosphorylation of fibroblast growth factor receptors KIRIN BEER KABUSHIKI KAISHA (JP) 2009-02-24 US disclosed
US-7495104-B2 Quinoline or quinazoline derivatives inhibiting auto-phosphorylation of fibroblast growth factor receptors KIRIN BEER KABUSHIKI KAISHA (JP) 2009-02-24 US disclosed