SCHEMBL13938233

SCHEMBL13938233

CCC(=O)OCCOc1ccc(-c2c(C#N)c(N)nc(SCc3csc(-c4ccc(Cl)cc4)n3)c2C#N)cc1

nearest known ligand 0.79

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 18/20 0.79
SLC6A3 Q01959 1/20 0.79
KDM4E B2RXH2 2/20 0.55
ALDH1A1 P00352 2/20 0.55
NPSR1 Q6W5P4 2/20 0.55
HSD17B10 Q99714 2/20 0.55
MEN1 O00255 1/20 0.55
POLB P06746 1/20 0.55
MAPT P10636 1/20 0.55
TSHR P16473 1/20 0.55
PPARG P37231 1/20 0.55
SMAD3 P84022 1/20 0.55
KMT2A Q03164 1/20 0.55
NCOA2 Q15596 1/20 0.55
NCOA1 Q15788 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
RXFP1 Q9HBX9 1/20 0.55
HPGD P15428 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3699454 0.93 ADORA1 (0.81) ADORA1SLC6A3KDM4EALDH1A1NPSR1
SCHEMBL1177362 0.93 ADORA1 (0.81) ADORA1SLC6A3
Hydrochloric Acid SCHEMBL3698557 0.92 ADORA1 (0.79) ADORA1SLC6A3KDM4EALDH1A1NPSR1
SCHEMBL13945016 0.92 ADORA1 (0.76) ADORA1SLC6A3KDM4EALDH1A1NPSR1
SCHEMBL7642574 0.92 ADORA1 (0.78) ADORA1SLC6A3KDM4EALDH1A1NPSR1
SCHEMBL3710188 0.91 ADORA1 (0.77) ADORA1SLC6A3KDM4EALDH1A1NPSR1
SCHEMBL13938560 0.91 ADORA1 (0.77) ADORA1SLC6A3
SCHEMBL13937445 0.91 ADORA1 (0.77) ADORA1SLC6A3
SCHEMBL3707223 0.90 ADORA1 (0.74) ADORA1SLC6A3KDM4EALDH1A1NPSR1
SCHEMBL3703461 0.90 ADORA1 (0.74) ADORA1SLC6A3KDM4EALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009015811-A1 DIPEPTOID PRODRUGS AND THE USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-02-05 WO disclosed