SCHEMBL13938245

SCHEMBL13938245

CC(C)CCn1c(O)c(C2=CS(=O)(=O)c3ccccc3N2)c(=O)n(CCC(C)C)c1=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.40
HSD17B10 Q99714 1/20 0.40
ALDH1A1 P00352 1/20 0.39
ADORA2A P29274 2/20 0.36
ADORA2B P29275 2/20 0.36
GAA P10253 1/20 0.34
PDE2A O00408 2/20 0.34
PDE1A P54750 1/20 0.34
PDE1B Q01064 1/20 0.34
PDE1C Q14123 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
THRB P10828 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
KDM4E B2RXH2 1/20 0.32
APAF1 O14727 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3930634 0.83 MAPK1 (0.55) MAPK1HSD17B10ALDH1A1GAACYP2C9
SCHEMBL13960689 0.82 MAPK1 (0.37) MAPK1HSD17B10GAACYP1A2CYP3A4
SCHEMBL7132364 0.80 MAPK1 (0.60) MAPK1HSD17B10ALDH1A1ADORA2AADORA2B
SCHEMBL3929186 0.80 MAPK1 (0.44) MAPK1HSD17B10ALDH1A1THRBRXFP1
SCHEMBL3918621 0.79 MAPK1 (0.44) MAPK1HSD17B10ALDH1A1CYP1A2CYP3A4
SCHEMBL3921269 0.77 MAPK1 (0.40) MAPK1HSD17B10ALDH1A1CYP2C9THRB
SCHEMBL7066378 0.76 MAPK1 (0.64) MAPK1HSD17B10ALDH1A1ADORA2AADORA2B
SCHEMBL7128338 0.76 MAPK1 (0.56) MAPK1HSD17B10ALDH1A1ADORA2AADORA2B
SCHEMBL7067237 0.74 MAPK1 (0.54) MAPK1HSD17B10ALDH1A1ADORA2AADORA2B
SCHEMBL7067024 0.74 MAPK1 (0.54) MAPK1HSD17B10ALDH1A1ADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7479489-B2 Heterocyclic antiviral compounds ROCHE PALO ALTO LLC (US) 2009-01-20 US disclosed