SCHEMBL13961608

SCHEMBL13961608

COBN1CCN(c2ccncc2NC(=O)c2ccnc(-c3cccc4sccc34)n2)CC1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 6/20 0.42
GSK3A P49840 3/20 0.42
GSK3B P49841 3/20 0.42
PIM1 P11309 6/20 0.41
PIM3 Q86V86 6/20 0.41
PIM2 Q9P1W9 5/20 0.39
ATR Q13535 3/20 0.39
HTR1A P08908 2/20 0.38
DRD2 P14416 2/20 0.38
HTR2A P28223 2/20 0.38
HTR2C P28335 1/20 0.37
ADRA1A P35348 1/20 0.37
HRH1 P35367 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13961711 0.90 CHEK1 (0.47) CHEK1GSK3AGSK3BPIM1PIM3
SCHEMBL13028325 0.86 GSK3B (0.44) CHEK1GSK3AGSK3BPIM1PIM3
SCHEMBL13027875 0.86 CHEK1 (0.55) CHEK1GSK3AGSK3BPIM1PIM3
SCHEMBL13067931 0.86 BACE1 (0.43) CHEK1GSK3AGSK3BPIM1PIM3
SCHEMBL13961449 0.85 GSK3B (0.42) CHEK1GSK3AGSK3BPIM1PIM3
SCHEMBL13961491 0.84 GSK3A (0.45) CHEK1GSK3AGSK3BPIM1PIM3
SCHEMBL13961490 0.84 CHEK1 (0.58) CHEK1GSK3AGSK3BPIM1PIM3
SCHEMBL13961609 0.83 GSK3B (0.46) CHEK1GSK3AGSK3BPIM1PIM3
SCHEMBL13961454 0.81 CHEK1 (0.56) CHEK1GSK3AGSK3BPIM1PIM3
SCHEMBL13961452 0.81 CHEK1 (0.45) CHEK1GSK3AGSK3BPIM1PIM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009014637-A2 HETEROCYCLIC AMIDE COMPOUNDS AS PROTEIN KINASE INHIBITORS SCHERING CORPORATION (US) 2009-01-29 WO disclosed