SCHEMBL1396237

SCHEMBL1396237

CS(=O)(=O)[Si](CCOCn1ccc2c(Cl)ncnc21)(S(C)(=O)=O)S(C)(=O)=O

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 2/20 0.35
FGFR4 P22455 2/20 0.35
SLC22A12 Q96S37 1/20 0.34
NOTUM Q6P988 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL98891 0.84 FGFR1 (0.35) FGFR1FGFR4SLC22A12
SCHEMBL18583995 0.83 FGFR1 (0.35) FGFR1FGFR4SLC22A12NOTUM
SCHEMBL18593997 0.78 FGFR1 (0.35) FGFR1FGFR4SLC22A12NOTUM
SCHEMBL10388320 0.77 TSHR (0.40) FGFR1FGFR4SLC22A12NOTUM
SCHEMBL29982155 0.76 FGFR1 (0.34) FGFR1FGFR4SLC22A12
SCHEMBL3003619 0.71 NOTUM (0.43) FGFR1FGFR4NOTUM
SCHEMBL31291523 0.71 NOTUM (0.43) FGFR1FGFR4NOTUM
SCHEMBL31720885 0.70 SLC22A12 (0.41) FGFR1FGFR4SLC22A12NOTUM
SCHEMBL1897615 0.70 SLC22A12 (0.41) FGFR1FGFR4SLC22A12NOTUM
SCHEMBL4255524 0.70 SLC22A12 (0.41) FGFR1FGFR4SLC22A12NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2288610-A1 AZETIDINE AND CYCLOBUTANE DERIVATIVES AS JAK INHIBITORS Incyte Corporation (US) 2011-03-02 EP disclosed
WO-2009114512-A1 AZETIDINE AND CYCLOBUTANE DERIVATIVES AS JAK INHIBITORS INCYTE CORPORATION (US) 2009-09-17 WO disclosed