SCHEMBL13972721

SCHEMBL13972721

CC1CN(c2c(F)c(F)c(NC(=O)C3CCC(N)CC3)c(F)c2F)CC(C)O1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.43
MAPK1 P28482 1/20 0.43
GSK3B P49841 3/20 0.36
MAPT P10636 2/20 0.36
POLB P06746 2/20 0.34
DYRK1A Q13627 2/20 0.33
WNT1 P04628 1/20 0.33
GAK O14976 1/20 0.33
BRAF P15056 1/20 0.33
KDR P35968 1/20 0.33
JAK2 O60674 2/20 0.32
JAK1 P23458 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
USP30 Q70CQ3 1/20 0.31
NPC1 O15118 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HSP90AB1 P08238 1/20 0.31
ULK1 O75385 1/20 0.31
SMYD3 Q9H7B4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13204150 0.81 NPY5R (0.45) TSHRMAPK1GSK3BMAPTPOLB
SCHEMBL10133397 0.81 NPY5R (0.45) TSHRMAPK1GSK3BMAPTPOLB
SCHEMBL10114350 0.81 NPY5R (0.45) TSHRMAPK1GSK3BMAPTPOLB
SCHEMBL14424161 0.81 NPY5R (0.45) TSHRMAPK1GSK3BMAPTPOLB
SCHEMBL10134102 0.80 TSHR (0.37) TSHRMAPK1GSK3BMAPTPOLB
SCHEMBL10114730 0.80 TSHR (0.37) TSHRMAPK1GSK3BMAPTPOLB
SCHEMBL13204301 0.80 TSHR (0.37) TSHRMAPK1GSK3BMAPTPOLB
SCHEMBL11941164 0.75 KDM4E (0.32)
SCHEMBL11935247 0.75 KDM4E (0.32)
SCHEMBL13438927 0.75 KDM4E (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2014285-A1 NPYY5 antagonists Shionogi&Co., Ltd. (JP) 2009-01-14 EP disclosed