SCHEMBL13985122

SCHEMBL13985122

C=C/C=C(\C=C/N)N1CCC2(CCN(C(=O)c3cccc(N4Cc5cccc(Cl)c5C4=O)c3)CC2)CC1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 1/20 0.66
CYP1A2 P05177 5/20 0.36
CYP3A4 P08684 5/20 0.36
USP2 O75604 3/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
MAPK1 P28482 2/20 0.36
ALDH1A1 P00352 4/20 0.36
TSHR P16473 2/20 0.36
CYP2D6 P10635 4/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 1/20 0.35
HIF1A Q16665 2/20 0.35
CHRM2 P08172 1/20 0.35
CHRM3 P20309 1/20 0.35
PARP1 P09874 2/20 0.35
EGFR P00533 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
GABRD O14764 1/20 0.34
GABRA1 P14867 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4716342 0.83 BDKRB1 (0.77) BDKRB1CYP1A2CYP3A4USP2MEN1
SCHEMBL4717762 0.81 BDKRB1 (0.74) BDKRB1CYP1A2CYP3A4USP2MEN1
SCHEMBL1712902 0.80 BDKRB1 (1.00) BDKRB1CYP1A2CYP3A4USP2MEN1
SCHEMBL4712523 0.80 BDKRB1 (0.72) BDKRB1CYP1A2CYP3A4USP2MEN1
SCHEMBL4714147 0.77 BDKRB1 (0.69) BDKRB1CYP1A2CYP3A4USP2MEN1
SCHEMBL4760693 0.76 BDKRB1 (0.66) BDKRB1USP2MAPK1ALDH1A1TSHR
SCHEMBL4716862 0.74 BDKRB1 (0.64) BDKRB1USP2MEN1KMT2AMAPK1
SCHEMBL4714259 0.73 BDKRB1 (0.60) BDKRB1MEN1KMT2AMAPK1ALDH1A1
SCHEMBL4759441 0.73 BDKRB1 (0.84) BDKRB1CYP1A2CYP3A4USP2MEN1
SCHEMBL4716396 0.73 BDKRB1 (0.61) BDKRB1MEN1KMT2APARP1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008153967-A1 BK1 ANTAGONIST CONJUGATES CONTEC THERAPEUTICS, INC. (US) 2008-12-18 WO disclosed