SCHEMBL13985779

SCHEMBL13985779

Cc1cc2c(s1)CN(C(=O)OC(C)(C)C)CC2

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.55
NR1H2 P55055 1/20 0.54
ADORA1 P30542 2/20 0.51
HDAC6 Q9UBN7 1/20 0.47
MAPT P10636 2/20 0.47
KDM4E B2RXH2 1/20 0.47
KCNQ2 O43526 1/20 0.45
MKNK1 Q9BUB5 7/20 0.43
MAPK1 P28482 1/20 0.42
GRAMD1A Q96CP6 1/20 0.41
BRD4 O60885 1/20 0.40
CREBBP Q92793 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6421569 0.89 ESR2 (0.55) ESR2NR1H2ADORA1HDAC6MAPT
SCHEMBL27141410 0.85 HDAC6 (0.58) ESR2NR1H2ADORA1HDAC6MAPT
SCHEMBL986037 0.85 ESR2 (0.54) ESR2NR1H2ADORA1HDAC6MAPT
SCHEMBL23142234 0.84 ESR2 (0.50) ESR2NR1H2ADORA1HDAC6MAPT
SCHEMBL976244 0.84 ADORA1 (0.55) ESR2NR1H2ADORA1HDAC6MAPT
SCHEMBL4815544 0.84 ESR2 (0.53) ESR2NR1H2ADORA1HDAC6MAPT
SCHEMBL27081538 0.83 HDAC6 (0.59) ESR2NR1H2ADORA1HDAC6MAPT
SCHEMBL13593457 0.83 ESR2 (0.52) ESR2NR1H2ADORA1HDAC6MAPT
SCHEMBL27141188 0.83 ESR2 (0.52) ESR2NR1H2ADORA1HDAC6MAPT
SCHEMBL13981293 0.83 ESR2 (0.52) ESR2NR1H2ADORA1HDAC6MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7468371-B2 Tricyclic pyrazole kinase inhibitors ABBOTT LABORATORIES INC. (US) 2008-12-23 US disclosed