SCHEMBL13986220

SCHEMBL13986220

CCc1cc(C)cc(-c2ccc3c(N)n[nH]c3c2)c1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.54
PDPK1 O15530 13/20 0.52
ABL1 P00519 2/20 0.50
BCR P11274 2/20 0.50
FGFR1 P11362 1/20 0.50
TGFBR1 P36897 6/20 0.49
AURKA O14965 5/20 0.49
AURKB Q96GD4 5/20 0.49
ROCK1 Q13464 3/20 0.49
SGK1 O00141 2/20 0.46
MKNK1 Q9BUB5 1/20 0.44
MKNK2 Q9HBH9 1/20 0.44
CHUK O15111 1/20 0.44
RPS6KB1 P23443 1/20 0.44
CDK2 P24941 1/20 0.44
KDR P35968 1/20 0.44
SYK P43405 1/20 0.44
JAK3 P52333 1/20 0.44
MAP3K5 Q99683 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13986221 0.87 PDPK1 (0.66) JAK2PDPK1ABL1BCRTGFBR1
SCHEMBL6478485 0.84 JAK2 (0.66) JAK2PDPK1ABL1BCRFGFR1
SCHEMBL13524482 0.83 JAK2 (0.50) JAK2PDPK1ABL1BCRFGFR1
SCHEMBL13525176 0.82 PDPK1 (0.65) JAK2PDPK1ABL1BCRTGFBR1
SCHEMBL13986219 0.80 JAK2 (0.56) JAK2PDPK1ABL1BCRFGFR1
SCHEMBL13525152 0.80 PDPK1 (0.57) JAK2PDPK1ABL1BCRTGFBR1
SCHEMBL6479941 0.79 JAK2 (0.72) JAK2PDPK1ABL1BCRTGFBR1
SCHEMBL4491663 0.78 PDPK1 (0.71) JAK2PDPK1ABL1BCRTGFBR1
SCHEMBL13524475 0.78 JAK2 (0.54) JAK2PDPK1ABL1BCRTGFBR1
SCHEMBL91579 0.77 PDPK1 (0.55) JAK2PDPK1FGFR1TGFBR1AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7459564-B2 Substituted biaryl compounds as factor XIa inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2008-12-02 US disclosed