SCHEMBL13993121

SCHEMBL13993121

COc1ccccc1-c1cc(N)n2ncc(Br)c2n1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 3/20 0.62
CHEK1 O14757 1/20 0.62
CCNA2 P20248 1/20 0.62
CCNA1 P78396 1/20 0.62
GSK3B P49841 4/20 0.48
HSP90AA1 P07900 2/20 0.48
HSP90AB1 P08238 1/20 0.47
KDM4E B2RXH2 3/20 0.46
ALDH1A1 P00352 3/20 0.46
MEN1 O00255 2/20 0.46
HPGD P15428 2/20 0.46
KMT2A Q03164 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
CSNK2A1 P68400 2/20 0.42
MAPT P10636 2/20 0.41
ADORA2A P29274 2/20 0.41
POLB P06746 1/20 0.41
GAA P10253 1/20 0.41
NPC1 O15118 1/20 0.40
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12953639 0.85 GSK3B (0.54) CDK2CHEK1CCNA2CCNA1GSK3B
SCHEMBL13993125 0.83 CDK2 (0.67) CDK2CHEK1CCNA2CCNA1GSK3B
SCHEMBL30579375 0.83 HSP90AA1 (0.46) CDK2CHEK1CCNA2CCNA1HSP90AA1
SCHEMBL12953613 0.81 CDK2 (0.67) CDK2CHEK1CCNA2CCNA1GSK3B
SCHEMBL12954497 0.81 GSK3B (0.67) CDK2CHEK1CCNA2CCNA1GSK3B
SCHEMBL13998512 0.78 GSK3B (0.62) CDK2GSK3BKDM4EALDH1A1MEN1
SCHEMBL14582875 0.78 GSK3B (0.72) CDK2CCNA2CCNA1GSK3BMEN1
SCHEMBL14607083 0.78 CDK2 (0.62) CDK2CHEK1CCNA2CCNA1GSK3B
SCHEMBL4177549 0.77 CDK2 (1.00) CDK2CHEK1CCNA2CCNA1GSK3B
SCHEMBL12953365 0.76 CDK2 (0.73) CDK2CCNA2CCNA1GSK3BMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7468372-B2 Trisubstituted 4-aminopyrazolopyrimidines as cyclin dependent kinase inhibitors SCHERING CORPORATION (US) 2008-12-23 US disclosed
US-7468372-B2 Trisubstituted 4-aminopyrazolopyrimidines as cyclin dependent kinase inhibitors SCHERING CORPORATION (US) 2008-12-23 US disclosed