SCHEMBL1399353

SCHEMBL1399353

COc1ccc2[nH]cc(Sc3cc(Cl)ccc3CCN)c2c1C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 10/20 0.45
TUBB4A P04350 3/20 0.45
TUBB P07437 3/20 0.45
TUBA3C P0DPH7 3/20 0.45
TUBA1B P68363 3/20 0.45
TUBA4A P68366 3/20 0.45
TUBB4B P68371 3/20 0.45
TUBB3 Q13509 3/20 0.45
TUBB2A Q13885 3/20 0.45
TUBB8 Q3ZCM7 3/20 0.45
TUBA3E Q6PEY2 3/20 0.45
TUBA1A Q71U36 3/20 0.45
TUBA1C Q9BQE3 3/20 0.45
TUBB6 Q9BUF5 3/20 0.45
TUBB2B Q9BVA1 3/20 0.45
TUBB1 Q9H4B7 3/20 0.45
HTR2A P28223 5/20 0.44
TRPM8 Q7Z2W7 2/20 0.43
CPT2 P23786 1/20 0.39
CPT1A P50416 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1399305 0.86 HTR2A (0.59) IDO1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL1399214 0.86 IDO1 (0.46) IDO1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL1399345 0.84 HTR2A (0.50) IDO1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL1399358 0.82 HTR2A (0.50) IDO1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL1399252 0.80 IDO1 (0.48) IDO1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL1399242 0.78 HTR2A (0.60) IDO1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL1399299 0.78 HTR2A (0.60) IDO1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL1399292 0.78 IDO1 (0.47) IDO1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL1399487 0.77 HTR2A (0.65) IDO1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL1399283 0.77 HTR2A (0.56) IDO1HTR2ATRPM8HTR1DCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1860100-B1 2-(1H-indolylsulfanyl)-benzyl amine derivatives as SSRI LUNDBECK & CO AS H (DK) 2011-03-02 EP claimed