SCHEMBL14015686

SCHEMBL14015686

CC(C)n1nc(-c2ccccc2)c(Cl)c1N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RET P07949 5/20 0.44
MERTK Q12866 1/20 0.43
RECQL P46063 1/20 0.42
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 2/20 0.42
GLA P06280 2/20 0.42
HPGD P15428 2/20 0.42
LMNA P02545 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
PDE1A P54750 1/20 0.41
PDE1B Q01064 1/20 0.41
PDE1C Q14123 1/20 0.41
KMT2A Q03164 1/20 0.40
KDR P35968 3/20 0.39
NPC1 O15118 1/20 0.39
GAA P10253 1/20 0.39
RAB9A P51151 1/20 0.39
ATM Q13315 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14015683 0.80 RET (0.44) RETMERTKSMN1; SMN2PDE1APDE1B
SCHEMBL13858455 0.77 MAPT (0.51) RECQLKDM4EALDH1A1GLAHPGD
SCHEMBL14015668 0.76 ESR1 (0.44) MERTKRECQLKDM4EALDH1A1PDE1A
SCHEMBL13858360 0.75 PDE1A (0.49) RETMERTKKDM4EALDH1A1GLA
SCHEMBL16200211 0.73 MEN1 (0.48) RECQLKDM4EALDH1A1GLAHPGD
SCHEMBL13715965 0.73 HTR2A (0.44) RETMERTKRECQLPDE1APDE1B
SCHEMBL13860832 0.72 NPC1 (0.51) KDM4EALDH1A1GLAHPGDLMNA
SCHEMBL17054305 0.70 PDE1A (0.51) RETMERTKRECQLKDM4EALDH1A1
SCHEMBL12377267 0.70 NPC1 (0.45) RETALDH1A1SMN1; SMN2PDE1APDE1B
SCHEMBL23402056 0.69 KMT2A (0.45) RETMERTKRECQLLMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7449576-B1 potent antagonists of the CCR1 receptor; inflammation; (5-Chloro-2-piperazin-1-yl-phenyl)-phenyl-methanone CHEMOCENTRYX, INC. (US) 2008-11-11 US disclosed