SCHEMBL14016397

SCHEMBL14016397

Bc1cc(C[C@@H](OC(=O)N2CCC(N3CCc4ccccc4NC3=O)CC2)C(=O)N2CCC(N3CCN(CC(=O)OCC)CC3)CC2)cc(B)c1O

nearest known ligand 0.68

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 20/20 0.68
RAMP1 O60894 2/20 0.68
CYP3A4 P08684 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14036254 0.96 CALCRL (0.64) CALCRLRAMP1CYP3A4
SCHEMBL14016666 0.94 CALCRL (0.63) CALCRLRAMP1CYP3A4
SCHEMBL2084967 0.93 CALCRL (0.78) CALCRLRAMP1CYP3A4
SCHEMBL2084965 0.93 CALCRL (0.78) CALCRLRAMP1CYP3A4
SCHEMBL14017778 0.92 CALCRL (0.63) CALCRLRAMP1CYP3A4
SCHEMBL2165222 0.92 CALCRL (0.68) CALCRLRAMP1CYP3A4
SCHEMBL2165231 0.92 CALCRL (0.68) CALCRLRAMP1CYP3A4
SCHEMBL2086979 0.92 CALCRL (0.77) CALCRLRAMP1CYP3A4
SCHEMBL2086981 0.92 CALCRL (0.77) CALCRLRAMP1CYP3A4
SCHEMBL14017749 0.91 CALCRL (0.66) CALCRLRAMP1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863791-B1 2-OXO-1,2,4,5-TETRAHYDRO-1,3-BENZODIAZEPIN-3-YL-PIPERIDINES USED AS CGRP ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2008-11-12 EP disclosed