SCHEMBL14016705

SCHEMBL14016705

C#Cc1cc(C[C@@H](CC(=O)N2CCC(N3Cc4ccccc4NC3=O)CC2)C(=O)N2CCC(N3CCCN(C)CC3)CC2)cc(Cl)c1N

nearest known ligand 0.67

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 20/20 0.67
RAMP1 O60894 1/20 0.67
CYP3A4 P08684 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14016949 0.97 CALCRL (0.70) CALCRLRAMP1CYP3A4
SCHEMBL14016941 0.95 CALCRL (0.67) CALCRLRAMP1CYP3A4
SCHEMBL14017258 0.95 CALCRL (0.63) CALCRLRAMP1CYP3A4
SCHEMBL14017084 0.94 CALCRL (0.75) CALCRLRAMP1CYP3A4
SCHEMBL14017151 0.94 CALCRL (0.64) CALCRLRAMP1CYP3A4
SCHEMBL14016844 0.94 CALCRL (0.70) CALCRLRAMP1CYP3A4
SCHEMBL14016703 0.92 CALCRL (0.79) CALCRLRAMP1CYP3A4
SCHEMBL14016950 0.92 CALCRL (0.61) CALCRLRAMP1CYP3A4
SCHEMBL14017137 0.91 CALCRL (0.61) CALCRLRAMP1CYP3A4
SCHEMBL14017127 0.91 CALCRL (0.61) CALCRLRAMP1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7439237-B2 Selected CGRP-antagonists, process for preparing them and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-10-21 US disclosed
US-7439237-B2 Selected CGRP-antagonists, process for preparing them and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-10-21 US disclosed