SCHEMBL14017167

SCHEMBL14017167

C#Cc1cc(C[C@@H](OC(=O)N2CCC(N3Cc4ccccc4NC3=O)CC2)C(=O)N2CCN(c3ccncc3)CC2)cc(Cl)c1N

nearest known ligand 0.52

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 20/20 0.52
RAMP1 O60894 4/20 0.51
CALCA P06881 1/20 0.49
CYP3A4 P08684 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14016968 0.94 CALCRL (0.58) CALCRLRAMP1CALCACYP3A4
SCHEMBL14017256 0.93 CALCRL (0.58) CALCRLRAMP1CALCA
SCHEMBL14017140 0.90 CALCRL (0.53) CALCRLRAMP1CALCACYP3A4
SCHEMBL14017143 0.89 CALCRL (0.53) CALCRLRAMP1CALCACYP3A4
SCHEMBL14375067 0.89 CALCRL (0.57) CALCRLRAMP1CYP3A4
SCHEMBL14017324 0.88 CALCRL (0.64) CALCRLRAMP1CYP3A4
SCHEMBL14017175 0.88 CALCRL (0.54) CALCRLRAMP1CALCA
SCHEMBL14016881 0.88 CALCRL (0.58) CALCRLRAMP1CYP3A4
SCHEMBL14016901 0.88 CALCRL (0.55) CALCRLRAMP1CYP3A4
SCHEMBL14017097 0.88 CALCRL (0.65) CALCRLRAMP1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7439237-B2 Selected CGRP-antagonists, process for preparing them and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-10-21 US disclosed