SCHEMBL14017757

SCHEMBL14017757

Bc1cc(C[C@@H](OC(=O)N2CCC(N3CCc4ccccc4NC3=O)CC2)C(=O)N2CCN(C3CCN(CC(=O)N(C)O)CC3)CC2)cc(C=C)c1O

nearest known ligand 0.60

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 19/20 0.60
RAMP1 O60894 2/20 0.60
CALCA P06881 1/20 0.38
CYP3A4 P08684 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14016426 0.98 CALCRL (0.60) CALCRLRAMP1CALCACYP3A4
SCHEMBL14017725 0.94 CALCRL (0.65) CALCRLRAMP1CALCACYP3A4
SCHEMBL14036286 0.91 CALCRL (0.62) CALCRLRAMP1CALCACYP3A4
SCHEMBL14017750 0.90 CALCRL (0.62) CALCRLRAMP1CYP3A4
SCHEMBL14017770 0.89 CALCRL (0.59) CALCRLRAMP1CYP3A4
SCHEMBL14016667 0.89 CALCRL (0.60) CALCRLRAMP1CALCACYP3A4
SCHEMBL14036221 0.89 CALCRL (0.61) CALCRLRAMP1CALCA
SCHEMBL14016979 0.89 CALCRL (0.60) CALCRLRAMP1CYP3A4
SCHEMBL2164959 0.89 CALCRL (0.66) CALCRLRAMP1CALCACYP3A4
SCHEMBL2166934 0.89 CALCRL (0.76) CALCRLRAMP1CALCACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863791-B1 2-OXO-1,2,4,5-TETRAHYDRO-1,3-BENZODIAZEPIN-3-YL-PIPERIDINES USED AS CGRP ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2008-11-12 EP disclosed