SCHEMBL1402141

SCHEMBL1402141

CCC(=O)N[C@H]1CC(n2cnc3c(NCC(c4ccccc4)c4ccccc4)nc(N4CC[C@@H](N)C4)nc32)C(O)[C@@H]1O

nearest known ligand 0.62

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 18/20 0.62
ADORA3 P0DMS8 10/20 0.62
CCNE2 O96020 1/20 0.46
CCNA2 P20248 1/20 0.46
CCNE1 P24864 1/20 0.46
CDK2 P24941 1/20 0.46
CCNA1 P78396 1/20 0.46
ADORA2B P29275 2/20 0.43
ADORA1 P30542 2/20 0.43
CDK1 P06493 1/20 0.42
CDK5 Q00535 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL239193 1.00 ADORA2A (0.62) ADORA2AADORA3CCNE2CCNA2CCNE1
SCHEMBL239194 1.00 ADORA2A (0.62) ADORA2AADORA3CCNE2CCNA2CCNE1
SCHEMBL1402143 1.00 ADORA2A (0.62) ADORA2AADORA3CCNE2CCNA2CCNE1
SCHEMBL13879042 1.00 ADORA2A (0.62) ADORA2AADORA3CCNE2CCNA2CCNE1
Hydrochloric Acid SCHEMBL2930221 0.99 ADORA2A (0.61) ADORA2AADORA3CCNE2CCNA2CCNE1
Hydrochloric Acid SCHEMBL1412246 0.99 ADORA2A (0.61) ADORA2AADORA3CCNE2CCNA2CCNE1
Hydrochloric Acid SCHEMBL2930224 0.99 ADORA2A (0.61) ADORA2AADORA3CCNE2CCNA2CCNE1
Hydrochloric Acid SCHEMBL1412250 0.99 ADORA2A (0.61) ADORA2AADORA3CCNE2CCNA2CCNE1
Trifluoroacetic Acid SCHEMBL2887186 0.96 ADORA2A (0.58) ADORA2AADORA3CCNE2CCNA2CCNE1
Hydrochloric Acid SCHEMBL1402112 0.95 ADORA2A (0.62) ADORA2AADORA3ADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2292619-A1 Purine derivatives for use as adenonsin A-2A receptor agonists Novartis AG (CH) 2011-03-09 EP disclosed