SCHEMBL14028482

SCHEMBL14028482

O=c1[nH]c(=O)c2c(C3CCCNC3)cc(-c3ccccc3O)nc2[nH]1

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 16/20 0.56
CHUK O15111 1/20 0.56
CDK1 P06493 1/20 0.39
CDK2 P24941 1/20 0.39
CHEK2 O96017 2/20 0.38
PRKCZ Q05513 1/20 0.37
PRKD2 Q9BZL6 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4942324 0.99 IKBKB (0.55) IKBKBCHUKCDK1CDK2CHEK2
SCHEMBL14028498 0.84 IKBKB (0.56) IKBKBCHUKCDK1CDK2CHEK2
Hydrochloric Acid SCHEMBL4944296 0.83 IKBKB (0.55) IKBKBCHUKCDK1CDK2CHEK2
SCHEMBL7197710 0.82 IKBKB (0.52) IKBKBCHUKCDK1CDK2CHEK2
Hydrochloric Acid SCHEMBL4945004 0.81 IKBKB (0.51) IKBKBCHUKCDK1CDK2CHEK2
SCHEMBL14028464 0.81 IKBKB (0.64) IKBKBCHUKCDK1CDK2
Hydrochloric Acid SCHEMBL4947782 0.80 IKBKB (0.63) IKBKBCHUKCDK1CDK2
SCHEMBL14028470 0.79 IKBKB (0.70) IKBKBCHUKCDK1CDK2CHEK2
Hydrochloric Acid SCHEMBL4945343 0.78 IKBKB (0.69) IKBKBCHUKCDK1CDK2CHEK2
SCHEMBL4942340 0.77 SMARCA2 (0.43) IKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7435743-B2 Pyridine derivatives BAYER AKTIENGESELLSCHAFT (DE) 2008-10-14 US disclosed
US-7435743-B2 Pyridine derivatives BAYER AKTIENGESELLSCHAFT (DE) 2008-10-14 US disclosed
US-7232909-B2 Pyridine derivatives BAYER AKTIENGESELLSCHAFT (DE) 2007-06-19 US disclosed
US-7232909-B2 Pyridine derivatives BAYER AKTIENGESELLSCHAFT (DE) 2007-06-19 US disclosed