SCHEMBL14040923

SCHEMBL14040923

O=C(c1cc2cnc(NC3CCOCC3)nc2s1)c1ccccc1O

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 10/20 0.42
MAPK3 P27361 3/20 0.42
SPR P35270 2/20 0.41
HDAC3 O15379 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
MAPK14 Q16539 6/20 0.40
LCK P06239 1/20 0.40
MAPK8 P45983 1/20 0.39
MAPK9 P45984 1/20 0.39
MAPK10 P53779 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4765914 0.89 MAPK14 (0.46) MAPK1MAPK3HDAC3HDAC1HDAC2
SCHEMBL4775106 0.89 MAPK14 (0.48) MAPK1MAPK3HDAC3HDAC1HDAC2
SCHEMBL14004218 0.87 HDAC3 (0.46) MAPK1MAPK3HDAC3HDAC1HDAC2
SCHEMBL14004217 0.76 MAPK8 (0.48) MAPK3MAPK8MAPK9MAPK10
SCHEMBL14004188 0.72 MAPK1 (0.49) MAPK1HDAC3HDAC1HDAC2HDAC6
SCHEMBL4771405 0.72 MAPK14 (0.43) MAPK1MAPK3HDAC3HDAC1HDAC2
SCHEMBL1517480 0.71 HDAC3 (0.45) MAPK1MAPK3HDAC3HDAC1HDAC2
SCHEMBL4765878 0.69 MAPK14 (0.59) MAPK1MAPK14LCKMAPK8MAPK9
SCHEMBL4776143 0.69 MAPK14 (0.44) MAPK1MAPK14LCKMAPK8MAPK9
SCHEMBL4776152 0.68 MAPK14 (0.53) MAPK1MAPK14MAPK8MAPK9MAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1485390-B1 BICYCLIC PYRIDINE AND PYRIMIDINE P38 KINASE INHIBITORS HOFFMANN LA ROCHE (CH) 2008-10-08 EP disclosed