SCHEMBL14048828

SCHEMBL14048828

Cc1c(Cc2cccc(N)n2)c(=O)oc2cc(OC(=O)N(C)C)c(I)cc12

nearest known ligand 0.61

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 20/20 0.61
RAF1 P04049 17/20 0.61
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL961051 0.89 MAP2K1 (0.72) MAP2K1RAF1
SCHEMBL959561 0.89 MAP2K1 (0.63) MAP2K1RAF1CYP3A4CYP2D6CYP2C9
SCHEMBL959933 0.84 MAP2K1 (0.71) MAP2K1RAF1CYP3A4CYP2C9
SCHEMBL959181 0.84 MAP2K1 (0.80) MAP2K1RAF1
SCHEMBL961264 0.78 MAP2K1 (0.85) MAP2K1RAF1CYP3A4CYP2C9
SCHEMBL960362 0.77 MAP2K1 (0.74) MAP2K1RAF1
SCHEMBL961410 0.77 MAP2K1 (0.83) MAP2K1RAF1CYP3A4CYP2C9
SCHEMBL961085 0.77 MAP2K1 (0.83) MAP2K1RAF1CYP3A4CYP2C9
SCHEMBL14048890 0.76 MAP2K1 (0.85) MAP2K1RAF1CYP3A4CYP2C9
SCHEMBL960164 0.76 MAP2K1 (1.00) MAP2K1RAF1CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1982982-A1 NOVEL COUMARIN DERIVATIVE HAVING ANTITUMOR ACTIVITY CHUGAI SEIYAKU KABUSHIKI KAISHA (JP) 2008-10-22 EP disclosed