SCHEMBL14064641

SCHEMBL14064641

Cc1ncn(-c2ccccc2CN)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NCF1 P14598 1/20 0.39
PDE9A O76083 1/20 0.39
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.33
PNMT P11086 1/20 0.33
LOXL2 Q9Y4K0 1/20 0.33
DPP4 P27487 2/20 0.32
TAAR1 Q96RJ0 1/20 0.32
SETDB1 Q15047 2/20 0.31
PSEN1 P49768 2/20 0.31
PSEN2 P49810 2/20 0.31
APH1B Q8WW43 2/20 0.31
NCSTN Q92542 2/20 0.31
APH1A Q96BI3 2/20 0.31
PSENEN Q9NZ42 2/20 0.31
CYP3A4 P08684 1/20 0.31
TNF P01375 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4832614 0.98 PDE9A (0.38) NCF1PDE9ACYP11B1CYP11B2LMNA
SCHEMBL4037271 0.78 DPP4 (0.33) DPP4PSEN1PSEN2APH1BNCSTN
SCHEMBL20455919 0.77 GAA (0.46) PDE9ALMNAMAPTSMN1; SMN2CYP3A4
Hydrochloric Acid SCHEMBL2076601 0.77 DPP4 (0.33) DPP4PSEN1PSEN2APH1BNCSTN
SCHEMBL16201996 0.77 FLT3 (0.44) CYP11B1CYP11B2LMNAMAPTSMN1; SMN2
SCHEMBL30332428 0.75 MAPT (0.47) NCF1PDE9AMAPTSMN1; SMN2PNMT
SCHEMBL8062086 0.75 MEN1 (0.43) MAPTSMN1; SMN2PSEN1PSEN2APH1B
SCHEMBL30725606 0.74 BCHE (0.40) LMNAMAPTSMN1; SMN2CYP3A4HCAR1
SCHEMBL12528439 0.74 BCHE (0.40) LMNAMAPTSMN1; SMN2CYP3A4HCAR1
SCHEMBL30725595 0.74 ADORA1 (0.47) LMNAMAPTSMN1; SMN2HCAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7419969-B2 HIV integrase inhibitors: cyclic pyrimidinone compounds BRISTOL-MYERS SQUIBB COMPANY (US) 2008-09-02 US disclosed
US-7419969-B2 HIV integrase inhibitors: cyclic pyrimidinone compounds BRISTOL-MYERS SQUIBB COMPANY (US) 2008-09-02 US disclosed
WO-2007058646-A1 HIV INTEGRASE INHIBITORS: CYCLIC PYRIMIDINONE COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-05-24 WO disclosed