SCHEMBL14067992

SCHEMBL14067992

CCS(=O)(=O)N(C)c1nc(C(=O)OC)c(O)c2ncc(C)cc12

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LCK P06239 1/20 0.34
ATM Q13315 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.31
RNASEH1 O60930 1/20 0.31
CYP2C9 P11712 1/20 0.31
THRB P10828 1/20 0.31
PIM3 Q86V86 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
PKM P14618 1/20 0.30
HPGD P15428 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4765621 0.81 KDM4E (0.43) KDM4EALDH1A1
SCHEMBL3969169 0.72 CYP19A1 (0.35) RNASEH1ALDH1A1HPGDNPSR1
SCHEMBL4072643 0.70 KDM4E (0.44) KDM4EALDH1A1
SCHEMBL4069766 0.69 ATM (0.41) LCKATMRNASEH1KDM4EALDH1A1
SCHEMBL27522607 0.64 ATM (0.44) ATMCYP2C9KDM4EALDH1A1HPGD
SCHEMBL31306918 0.62 ATM (0.53) LCKATMKDM4EALDH1A1HPGD
SCHEMBL24661703 0.61 ATM (0.47) ATMKDM4EALDH1A1PKMNPSR1
SCHEMBL3891700 0.61 GRM2 (0.41) RNASEH1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL31347580 0.61 ATM (0.50) ATMKDM4EALDH1A1NPSR1HSD17B10
SCHEMBL8272321 0.61 ATM (0.50) ATMKDM4EALDH1A1NPSR1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1496836-B1 N-(SUBSTITUTED BENZYL)-8-HYDROXY-1,6-NAPHTHYRIDINE-7- CARBOXAMIDES USEFUL AS HIV INTEGRASE INHIBITORS MERCK & CO INC (US) 2008-09-24 EP disclosed