SCHEMBL14068432

SCHEMBL14068432

Cc1cncc(OC[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C)c1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.54
ACE P12821 1/20 0.47
CYP3A4 P08684 5/20 0.47
APP P05067 4/20 0.46
CTSS P25774 2/20 0.44
CTSL P07711 1/20 0.44
CTSB P07858 1/20 0.44
CTSK P43235 1/20 0.44
JAK2 O60674 1/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
PKM P14618 1/20 0.42
HPGD P15428 1/20 0.42
HTT P42858 1/20 0.42
KMT2A Q03164 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
KLK5 Q9Y337 1/20 0.42
SYK P43405 1/20 0.41
PPARA Q07869 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6857744 0.89 ATM (0.53) ATMACECYP3A4APPCTSS
SCHEMBL14030166 0.89 ATM (0.53) ATMACECYP3A4APPCTSS
SCHEMBL6857746 0.89 ATM (0.53) ATMACECYP3A4APPCTSS
SCHEMBL14004830 0.89 ATM (0.53) ATMACECYP3A4APPCTSS
SCHEMBL14068584 0.88 ATM (0.39) ATMACECYP3A4JAK2ALDH1A1
SCHEMBL6854766 0.87 ATM (0.51) ATMACECYP3A4APPCTSS
SCHEMBL6854769 0.87 ATM (0.51) ATMACECYP3A4APPCTSS
SCHEMBL30639552 0.84 ATM (0.65) ATMACECYP3A4APPCTSS
SCHEMBL7596617 0.81 ATM (0.51) ATMACECYP3A4APP
SCHEMBL14441492 0.81 ATM (0.51) ATMACECYP3A4APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008109613-A1 BENZO[C][2,7]NAPHTHYRIDINE DERIVATIVES, AND THEIR USE AS KINASE INHIBITORS WYETH (US) 2008-09-12 WO disclosed