SCHEMBL14069857

SCHEMBL14069857

Cc1ccc(C(=O)Nc2cccc(C(F)(F)F)c2)cc1Nc1nn(C)c2nc(NCCCN(C)C)ncc12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 5/20 0.58
BRAF P15056 10/20 0.56
LCK P06239 6/20 0.56
KDR P35968 4/20 0.56
INSR P06213 4/20 0.56
LYN P07948 4/20 0.56
HCK P08631 4/20 0.56
SRC P12931 4/20 0.56
ESYT2 A0FGR8 2/20 0.56
NBAS A2RRP1 2/20 0.56
CNOT1 A5YKK6 2/20 0.56
TBKBP1 A7MCY6 2/20 0.56
AGPS O00116 2/20 0.56
MYO1F O00160 2/20 0.56
SNAP23 O00161 2/20 0.56
AP3B1 O00203 2/20 0.56
PSMD12 O00232 2/20 0.56
BMPR1B O00238 2/20 0.56
PGRMC1 O00264 2/20 0.56
CLIC1 O00299 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14069863 0.98 BTK (0.58) BTKBRAFLCKKDRINSR
SCHEMBL14070282 0.96 BTK (0.60) BTKBRAFLCKKDRINSR
SCHEMBL14070189 0.92 BTK (0.65) BTKBRAFLCKKDRINSR
SCHEMBL14070248 0.92 BTK (0.60) BTKBRAFLCKKDRINSR
SCHEMBL14070275 0.91 BTK (0.59) BTKBRAFLCKKDRINSR
SCHEMBL14069836 0.90 BTK (0.67) BTKBRAFLCKKDRINSR
SCHEMBL14070271 0.90 BTK (0.61) BTKBRAFLCKKDRINSR
SCHEMBL14070277 0.89 BTK (0.60) BTKBRAFLCKKDRINSR
SCHEMBL14069856 0.89 LCK (0.66) BTKBRAFLCKKDRINSR
SCHEMBL14070219 0.87 BTK (0.56) BTKBRAFLCKKDRINSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008112695-A2 PYRAZOLO [3,4-D] PYRIMIDINES AND 1, 2, 5, 6-TETRAAZA- AS- INDACENES AS PROTEIN KINASE INHIBITORS FOR CANCER TREATMENT IRM LLC (BM) 2008-09-18 WO disclosed