SCHEMBL14070901

SCHEMBL14070901

COc1ccc2c(c1)[C@H](C)[C@@](C)(C(=O)O)Cn1c-2c(C2CCCCC2)c2ccc(C(=O)NS(=O)(=O)N(C)C)cc21

nearest known ligand 0.67

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 10/20 0.67
KCNH2 Q12809 7/20 0.67
CYP3A4 P08684 3/20 0.66
SCN5A Q14524 2/20 0.66
CYP2C9 P11712 1/20 0.62
CYP2C19 P33261 1/20 0.62
SCN9A Q15858 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14342822 1.00 NR1I2 (0.67) NR1I2KCNH2CYP3A4SCN5ACYP2C9
SCHEMBL13846669 0.94 NR1I2 (0.60) NR1I2KCNH2CYP3A4SCN5ACYP2C9
SCHEMBL13841553 0.92 KCNH2 (0.57) NR1I2KCNH2CYP3A4SCN5ACYP2C9
SCHEMBL14095053 0.91 NR1I2 (0.68) NR1I2KCNH2CYP3A4SCN5ACYP2C9
SCHEMBL14026076 0.90 NR1I2 (0.67) NR1I2KCNH2CYP3A4SCN5ACYP2C9
SCHEMBL14095546 0.90 NR1I2 (0.62) NR1I2KCNH2CYP3A4SCN5ACYP2C9
SCHEMBL16711671 0.90 NR1I2 (0.81) NR1I2KCNH2CYP3A4SCN5ACYP2C9
SCHEMBL18051484 0.90 NR1I2 (0.56) NR1I2KCNH2CYP3A4SCN5ACYP2C9
SCHEMBL10155794 0.89 KCNH2 (0.55) NR1I2KCNH2CYP3A4SCN5ACYP2C9
SCHEMBL14343917 0.89 NR1I2 (0.64) NR1I2KCNH2CYP3A4SCN5ACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2118109-B1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL MYERS SQUIBB CO (US) 2014-11-26 EP disclosed
WO-2008112473-A1 COMPOUNDS FOR THE TREATMENT OF HEPATITIS C BRISTOL-MYERS SQUIBB COMPANY (US) 2008-09-18 WO disclosed