SCHEMBL1407943

SCHEMBL1407943

Cc1ncoc1-c1nnc(SCCCN2C[C@@H]3C[C@@]3(c3ccc(C(F)(F)F)cc3F)C2)n1C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 20/20 1.00
KCNH2 Q12809 19/20 1.00
DRD2 P14416 14/20 1.00
DRD4 P21917 1/20 1.00
CYP1A2 P05177 1/20 0.79
CYP2C19 P33261 1/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3243567 1.00 DRD3 (1.00) DRD3KCNH2DRD2DRD4CYP1A2
SCHEMBL13079532 1.00 DRD3 (1.00) DRD3KCNH2DRD2DRD4CYP1A2
SCHEMBL1407749 1.00 DRD3 (1.00) DRD3KCNH2DRD2DRD4CYP1A2
SCHEMBL3980374 1.00 DRD3 (1.00) DRD3KCNH2DRD2DRD4CYP1A2
SCHEMBL1407940 1.00 DRD3 (1.00) DRD3KCNH2DRD2DRD4CYP1A2
Hydrochloric Acid SCHEMBL1407735 0.99 DRD3 (0.98) DRD3KCNH2DRD2DRD4CYP1A2
Hydrochloric Acid SCHEMBL4259820 0.99 DRD3 (0.98) DRD3KCNH2DRD2DRD4CYP1A2
SCHEMBL11914910 0.94 DRD3 (1.00) DRD3KCNH2DRD2DRD4CYP1A2
SCHEMBL12313275 0.94 DRD3 (1.00) DRD3KCNH2DRD2DRD4CYP1A2
SCHEMBL378184 0.94 DRD3 (1.00) DRD3KCNH2DRD2DRD4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1917013-B1 USE OF AZABICYCLO HEXANE DERIVATIVES GLAXO GROUP LTD (GB) 2011-03-09 EP claimed
EP-1745040-B9 AZABICYCLO(3.1.0) HEXANE DERIVATIVES USEFUL AS MODULATORS OF DOPAMINE D3 RECEPTORS GLAXO GROUP LTD (GB) 2010-06-02 EP claimed
EP-1745040-B1 AZABICYCLO(3.1.0) HEXANE DERIVATIVES USEFUL AS MODULATORS OF DOPAMINE D3 RECEPTORS GLAXO GROUP LTD (GB) 2009-12-09 EP claimed