SCHEMBL14099208

SCHEMBL14099208

CC(=O)c1cc(-c2ccc(C(N)=O)c(Cl)c2)cc2c1OCCCC2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.40
MKNK1 Q9BUB5 1/20 0.39
MKNK2 Q9HBH9 1/20 0.39
NOTUM Q6P988 1/20 0.35
RORC P51449 1/20 0.35
PDK2 Q15119 1/20 0.34
JAK2 O60674 3/20 0.34
JAK1 P23458 2/20 0.34
TYK2 P29597 2/20 0.34
JAK3 P52333 2/20 0.34
KMT2A Q03164 2/20 0.33
KDM4E B2RXH2 2/20 0.33
LMNA P02545 2/20 0.33
PIK3CD O00329 1/20 0.33
ABL1 P00519 1/20 0.33
EGFR P00533 1/20 0.33
HCK P08631 1/20 0.33
SRC P12931 1/20 0.33
KDR P35968 1/20 0.33
PIK3CA P42336 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4643990 0.90 PARP1 (0.40) PARP1MKNK1MKNK2NOTUMRORC
SCHEMBL14161471 0.87 KDM4E (0.38) NOTUMPDK2KMT2AKDM4ELMNA
SCHEMBL4642110 0.78 KDM4E (0.40) NOTUMPDK2KMT2AKDM4ELMNA
SCHEMBL4640368 0.75 NOTUM (0.39) NOTUMPDK2KMT2AKDM4ELMNA
SCHEMBL4640367 0.74 HTT (0.48) RORCJAK2JAK1TYK2JAK3
SCHEMBL4736986 0.71 MKNK1 (0.43) MKNK1MKNK2PDK2KMT2AKDM4E
SCHEMBL3945829 0.70 KDM4E (0.45) KDM4ELMNAALDH1A1HSD17B10
SCHEMBL3935043 0.70 MAPK1 (0.42) KMT2AKDM4ELMNAMAPTHTT
SCHEMBL14161476 0.69 PARP1 (0.40) PARP1PIK3CAALDH1A1
SCHEMBL14098995 0.68 PARP1 (0.53) PARP1RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1956016-A1 Bicyclic acyltryptophanols Bayer Schering Pharma Aktiengesellschaft (DE) 2008-08-13 EP disclosed