SCHEMBL14101032

SCHEMBL14101032

CC(C)(C)OC(=O)N1CCc2c(N)cc(C(F)(F)F)cc2C1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.55
ESR2 Q92731 1/20 0.50
ADORA1 P30542 2/20 0.46
MAPT P10636 3/20 0.43
KDM4E B2RXH2 1/20 0.43
STS P08842 1/20 0.43
MAPK1 P28482 1/20 0.41
TACR1 P25103 1/20 0.39
F12 P00748 2/20 0.38
RAF1 P04049 1/20 0.38
BRAF P15056 1/20 0.38
JAK2 O60674 1/20 0.38
JAK3 P52333 1/20 0.38
PTK2 Q05397 1/20 0.38
UCHL1 P09936 1/20 0.38
SCN9A Q15858 1/20 0.38
GPR119 Q8TDV5 1/20 0.38
LIPG Q9Y5X9 1/20 0.37
ABHD6 Q9BV23 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30752205 0.87 NR1H2 (0.52) NR1H2ESR2ADORA1MAPTKDM4E
SCHEMBL27042717 0.87 NR1H2 (0.52) NR1H2ESR2ADORA1MAPTKDM4E
SCHEMBL13650434 0.84 ESR2 (0.48) NR1H2ESR2ADORA1MAPTKDM4E
SCHEMBL27042578 0.83 NR1H2 (0.57) NR1H2ESR2ADORA1MAPTKDM4E
SCHEMBL30752212 0.83 NR1H2 (0.57) NR1H2ESR2ADORA1MAPTKDM4E
SCHEMBL13645895 0.83 ESR2 (0.47) NR1H2ESR2ADORA1MAPTSTS
SCHEMBL14101081 0.81 ESR1 (0.49) ESR2KDM4EABHD6
SCHEMBL394214 0.80 NR1H2 (0.60) NR1H2ESR2ADORA1MAPTKDM4E
SCHEMBL29526229 0.80 NR1H2 (0.60) NR1H2ESR2ADORA1MAPTKDM4E
SCHEMBL19684693 0.80 ESR2 (0.54) NR1H2ESR2ADORA1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501803-B1 TETRAHYDROPYRANYL CYCLOPENTYL TETRAHYDROISOQUINOLINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO INC (US) 2008-08-13 EP disclosed