SCHEMBL14102012

SCHEMBL14102012

CN(C)C(=O)c1ccc(-n2nc(-c3ccccc3)c3ccccc3c2=O)c([N+](=O)O)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 5/20 0.49
MAPT P10636 4/20 0.49
GAA P10253 3/20 0.49
LMNA P02545 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.47
HTT P42858 3/20 0.46
HPGD P15428 3/20 0.46
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
HTR6 P50406 1/20 0.46
NCOA1 Q15788 1/20 0.43
NCOA3 Q9Y6Q9 1/20 0.43
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
ALOX15 P16050 1/20 0.41
ALOX5 P09917 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4723874 0.91 MAPT (0.59) NPSR1MAPTGAALMNASMN1; SMN2
SCHEMBL4723638 0.84 MAPT (0.67) NPSR1MAPTGAALMNASMN1; SMN2
SCHEMBL14102013 0.81 NPSR1 (0.54) NPSR1MAPTGAALMNASMN1; SMN2
SCHEMBL14102065 0.81 NPSR1 (0.58) NPSR1MAPTGAALMNASMN1; SMN2
SCHEMBL4720311 0.80 MAPT (0.63) NPSR1MAPTGAALMNAHTT
SCHEMBL4722447 0.78 MAPT (0.61) NPSR1MAPTGAALMNASMN1; SMN2
SCHEMBL4719235 0.75 MAPT (0.55) NPSR1MAPTGAALMNASMN1; SMN2
SCHEMBL14102062 0.75 NPSR1 (0.59) NPSR1MAPTGAALMNASMN1; SMN2
SCHEMBL4721037 0.73 NPSR1 (0.72) NPSR1MAPTGAALMNAHTT
SCHEMBL4721601 0.72 MAPT (0.70) NPSR1MAPTGAALMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed