SCHEMBL1410667

SCHEMBL1410667

C/C(=C\c1ccc(C)nc1)C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.53
TBXAS1 P24557 10/20 0.51
MAPT P10636 2/20 0.41
ALDH1A1 P00352 1/20 0.41
KDM4E B2RXH2 1/20 0.40
TSHR P16473 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
S1PR4 O95977 1/20 0.39
LMNA P02545 1/20 0.39
S1PR1 P21453 1/20 0.39
MAPK1 P28482 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
APEX1 P27695 1/20 0.38
HTT P42858 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1410669 1.00 AKR1C3 (0.53) AKR1C3TBXAS1MAPTALDH1A1KDM4E
SCHEMBL17188865 0.84 HDAC1 (0.41) TBXAS1MAPTALDH1A1KDM4ETSHR
SCHEMBL10992573 0.83 AKR1C3 (0.47) AKR1C3TBXAS1MAPTALDH1A1KMT2A
SCHEMBL10992577 0.83 AKR1C3 (0.47) AKR1C3TBXAS1MAPTALDH1A1KMT2A
SCHEMBL17368452 0.82 AKR1C3 (0.53) AKR1C3TBXAS1ALDH1A1KDM4EAPEX1
SCHEMBL17273936 0.82 AKR1C3 (0.53) AKR1C3TBXAS1APEX1
SCHEMBL2272168 0.81 AKR1C3 (0.52) AKR1C3TBXAS1ALDH1A1KDM4ESMN1; SMN2
SCHEMBL15758231 0.81 AKR1C3 (0.52) AKR1C3TBXAS1ALDH1A1MEN1KMT2A
SCHEMBL2272174 0.81 AKR1C3 (0.52) AKR1C3TBXAS1ALDH1A1KDM4ESMN1; SMN2
SCHEMBL15758230 0.81 AKR1C3 (0.52) AKR1C3TBXAS1ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2295410-A1 HDAC inhibitor Chroma Therapeutics Limited (GB) 2011-03-16 EP disclosed