SCHEMBL14106964

SCHEMBL14106964

CC(=O)N1c2ncccc2NC2=C(C(=O)CC(C)(C)C2)[C@@H]1c1ccc(OCc2ccccc2)c(Cl)c1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.49
KMT2A Q03164 4/20 0.49
KDM4E B2RXH2 4/20 0.45
NPC1 O15118 1/20 0.42
PTGES O14684 1/20 0.41
ALOX5 P09917 1/20 0.41
ALDH1A1 P00352 3/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 4/20 0.40
HPGD P15428 2/20 0.39
CASP1 P29466 2/20 0.39
CASP7 P55210 2/20 0.39
USP2 O75604 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14107086 1.00 MEN1 (0.49) MEN1KMT2AKDM4ENPC1PTGES
SCHEMBL13704068 0.89 MEN1 (0.62) MEN1KMT2AKDM4ENPC1PTGES
SCHEMBL13704070 0.89 MEN1 (0.62) MEN1KMT2AKDM4ENPC1PTGES
SCHEMBL4294419 0.89 MEN1 (0.62) MEN1KMT2AKDM4ENPC1PTGES
SCHEMBL14582940 0.84 MEN1 (0.53) MEN1KMT2AKDM4ENPC1PTGES
SCHEMBL14103352 0.82 MEN1 (0.49) MEN1KMT2AKDM4ENPC1PTGES
SCHEMBL14103362 0.82 MEN1 (0.49) MEN1KMT2AKDM4ENPC1PTGES
SCHEMBL14103364 0.82 MEN1 (0.49) MEN1KMT2AKDM4ENPC1PTGES
SCHEMBL13704066 0.80 MEN1 (0.72) MEN1KMT2AKDM4ENPC1ALDH1A1
SCHEMBL4289448 0.80 MEN1 (0.67) MEN1KMT2AKDM4EALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008099021-A1 DIBENZODIAZEPINONES USEFUL AS HEPATITIS C VIRUS INHIBITORS TIBOTEC PHARMACEUTICALS LTD. (IE) 2008-08-21 WO disclosed