SCHEMBL14106967

SCHEMBL14106967

CC(=O)N1c2ncncc2NC2=C(C(=O)CC(C)(C)C2)C1c1ccc(Cl)cc1Cl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.45
KMT2A Q03164 3/20 0.45
HSD17B10 Q99714 3/20 0.41
ALDH1A1 P00352 5/20 0.41
KDM4E B2RXH2 2/20 0.40
MAPT P10636 2/20 0.38
GSK3A P49840 2/20 0.37
GSK3B P49841 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
GAA P10253 3/20 0.37
GLA P06280 2/20 0.37
HPGD P15428 1/20 0.36
FPR1 P21462 1/20 0.36
MAPK13 O15264 1/20 0.36
DAPK3 O43293 1/20 0.36
ROCK2 O75116 1/20 0.36
CHEK2 O96017 1/20 0.36
PIM1 P11309 1/20 0.36
CDK2 P24941 1/20 0.36
RECQL P46063 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14107088 0.86 MEN1 (0.48) MEN1KMT2AHSD17B10ALDH1A1KDM4E
SCHEMBL14107085 0.86 MEN1 (0.48) MEN1KMT2AHSD17B10ALDH1A1KDM4E
SCHEMBL4744098 0.86 MEN1 (0.48) MEN1KMT2AHSD17B10ALDH1A1KDM4E
SCHEMBL14107072 0.84 HSD17B10 (0.41) MEN1KMT2AHSD17B10ALDH1A1KDM4E
SCHEMBL4291113 0.83 MEN1 (0.49) MEN1KMT2AHSD17B10ALDH1A1KDM4E
SCHEMBL4287691 0.82 MEN1 (0.62) MEN1KMT2AHSD17B10ALDH1A1KDM4E
SCHEMBL4290980 0.81 MEN1 (0.48) MEN1KMT2AHSD17B10ALDH1A1KDM4E
SCHEMBL4296680 0.80 MEN1 (0.47) MEN1KMT2AHSD17B10ALDH1A1MAPT
SCHEMBL13704059 0.80 MEN1 (0.48) MEN1KMT2AHSD17B10ALDH1A1KDM4E
SCHEMBL4287067 0.79 MEN1 (0.48) MEN1KMT2AHSD17B10ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008099021-A1 DIBENZODIAZEPINONES USEFUL AS HEPATITIS C VIRUS INHIBITORS TIBOTEC PHARMACEUTICALS LTD. (IE) 2008-08-21 WO disclosed