SCHEMBL14126747

SCHEMBL14126747

NC(=O)c1cc(Cl)cc2cc(C(=O)O)c(=O)[nH]c12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.46
HPGD P15428 3/20 0.40
HSD17B10 Q99714 3/20 0.40
POLB P06746 2/20 0.40
GPR35 Q9HC97 2/20 0.40
USP2 O75604 1/20 0.40
ALOX15 P16050 1/20 0.40
ALOX12 P18054 1/20 0.40
CASP1 P29466 1/20 0.40
CASP7 P55210 1/20 0.40
CYP3A4 P08684 1/20 0.40
KDM4E B2RXH2 5/20 0.39
GAA P10253 3/20 0.39
ALDH1A1 P00352 3/20 0.38
AKR1C4 P17516 1/20 0.38
AKR1C3 P42330 1/20 0.38
AKR1C2 P52895 1/20 0.38
AKR1C1 Q04828 1/20 0.38
PKM P14618 1/20 0.37
CYP1A2 P05177 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2310258 0.80 KDM4E (0.51) DYRK1AHPGDHSD17B10POLBGPR35
SCHEMBL14126859 0.79 DYRK1A (0.41) DYRK1AHPGDHSD17B10POLBGPR35
Bromide SCHEMBL14126727 0.78 DYRK1A (0.40) DYRK1AHPGDHSD17B10POLBGPR35
Hydrochloric Acid SCHEMBL14126717 0.78 DYRK1A (0.40) DYRK1AHPGDHSD17B10POLBGPR35
SCHEMBL14126724 0.77 KDM4E (0.39) DYRK1AHPGDHSD17B10POLBGPR35
SCHEMBL14126852 0.77 KDM4E (0.39) DYRK1AHPGDHSD17B10POLBGPR35
SCHEMBL14126594 0.77 DYRK1A (0.39) DYRK1AHPGDHSD17B10POLBGPR35
SCHEMBL14126723 0.77 KDM4E (0.39) DYRK1AHPGDHSD17B10POLBGPR35
SCHEMBL14126998 0.77 DYRK1A (0.41) DYRK1AHPGDHSD17B10POLBGPR35
SCHEMBL20559286 0.77 CNR2 (0.53) DYRK1AHPGDHSD17B10POLBGPR35

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012164085-A1 GLYCINE B ANTAGONISTS MERZ PHARMA GMBH & CO. KGAA (DE) 2012-12-06 WO claimed
WO-2012164085-A1 GLYCINE B ANTAGONISTS MERZ PHARMA GMBH & CO. KGAA (DE) 2012-12-06 WO disclosed