SCHEMBL14129459

SCHEMBL14129459

O=S(=O)(c1ccccc1)n1cccc1CNCc1ccc(CN(Cc2nc3ccccc3[nH]2)C2CCCc3cccnc32)cc1

nearest known ligand 0.69

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 20/20 0.69
CHRM2 P08172 1/20 0.54
CYP2D6 P10635 1/20 0.54
DRD2 P14416 1/20 0.54
OPRM1 P35372 1/20 0.54
KCNH2 Q12809 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4064574 0.95 CXCR4 (0.66) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL4061430 0.87 CXCR4 (0.75) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL4069793 0.87 CXCR4 (0.87) CXCR4CHRM2CYP2D6DRD2OPRM1
Bromide SCHEMBL5140353 0.86 CXCR4 (0.86) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL4063485 0.85 CXCR4 (0.87) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL4065687 0.85 CXCR4 (0.71) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL4069312 0.84 CXCR4 (0.86) CXCR4CHRM2CYP2D6DRD2OPRM1
Bromide SCHEMBL5140052 0.84 CXCR4 (0.86) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL4073962 0.84 CXCR4 (0.84) CXCR4CHRM2CYP2D6DRD2OPRM1
SCHEMBL4069614 0.83 CXCR4 (0.78) CXCR4CHRM2CYP2D6DRD2OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7396840-B2 Chemokine receptor binding heterocyclic compounds GENZYME CORPORATION (US) 2008-07-08 US disclosed
US-7396840-B2 Chemokine receptor binding heterocyclic compounds GENZYME CORPORATION (US) 2008-07-08 US disclosed