SCHEMBL14136752

SCHEMBL14136752

O=C(O)C1=CC2(CCC1S(=O)(=O)Nc1ccc(F)cc1Br)OC(CO)C(CO)O2

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TLR4 O00206 5/20 0.37
METAP2 P50579 3/20 0.31
MRGPRX1 Q96LB2 2/20 0.31
TSPO P30536 1/20 0.31
NPC1 O15118 1/20 0.30
MAPT P10636 1/20 0.30
PKM P14618 1/20 0.30
RAB9A P51151 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4154953 1.00 TLR4 (0.37) TLR4METAP2MRGPRX1TSPONPC1
SCHEMBL15093757 1.00 TLR4 (0.37) TLR4METAP2MRGPRX1TSPONPC1
SCHEMBL4163042 1.00 TLR4 (0.37) TLR4METAP2MRGPRX1TSPONPC1
SCHEMBL4153932 0.91 TLR4 (0.38) TLR4NPC1RAB9ASMN1; SMN2
SCHEMBL17727702 0.91 TLR4 (0.38) TLR4NPC1RAB9ASMN1; SMN2
SCHEMBL4145794 0.91 TLR4 (0.38) TLR4NPC1RAB9ASMN1; SMN2
SCHEMBL17727727 0.89 TLR4 (0.49) TLR4MRGPRX1NPC1PKMRAB9A
SCHEMBL14136690 0.89 TLR4 (0.49) TLR4MRGPRX1NPC1PKMRAB9A
SCHEMBL4141115 0.89 TLR4 (0.49) TLR4MRGPRX1NPC1PKMRAB9A
SCHEMBL4146514 0.89 TLR4 (0.49) TLR4MRGPRX1NPC1PKMRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1935879-B1 SUBSTITUTED CYCLOALKENE DERIVATIVE DAIICHI SANKYO CO LTD (JP) 2016-05-11 EP claimed
US-RE43858-E1 Substituted cycloalkene derivative DAIICHI SANKYO COMPANY, LIMITED (JP) 2012-12-11 US claimed