SCHEMBL14178951

SCHEMBL14178951

CC(=O)c1ccc(C#CCNC(=O)c2cc3cc(OCCN(C)C)ccc3[nH]2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 2/20 0.54
PDGFRA P16234 2/20 0.54
FLT3 P36888 1/20 0.52
HRH3 Q9Y5N1 2/20 0.45
HRH4 Q9H3N8 1/20 0.45
HTR2C P28335 1/20 0.42
KDM4E B2RXH2 6/20 0.42
ALDH1A1 P00352 3/20 0.42
MAPT P10636 3/20 0.42
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
RXFP1 Q9HBX9 1/20 0.41
SYK P43405 2/20 0.40
PYGL P06737 1/20 0.40
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
DRD2 P14416 1/20 0.39
DRD3 P35462 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4821303 0.92 PDGFRB (0.53) PDGFRBPDGFRAFLT3HRH3HRH4
SCHEMBL4818482 0.92 PDGFRB (0.53) PDGFRBPDGFRAFLT3HRH3HRH4
Hydrochloric Acid SCHEMBL4815345 0.91 PDGFRB (0.52) PDGFRBPDGFRAFLT3HRH3HRH4
SCHEMBL14613774 0.90 PDGFRB (0.52) PDGFRBPDGFRAFLT3HRH3HRH4
SCHEMBL14178952 0.90 KDM4E (0.46) PDGFRBPDGFRAFLT3KDM4EALDH1A1
SCHEMBL4250060 0.90 PDGFRB (0.51) PDGFRBPDGFRAFLT3HRH3HRH4
SCHEMBL8312368 0.81 HDAC1 (0.46) KDM4EALDH1A1MAPTNPC1RAB9A
SCHEMBL14613790 0.81 KDM4E (0.46) KDM4EALDH1A1MAPTNPC1RAB9A
SCHEMBL15223791 0.79 PDGFRB (0.74) PDGFRBPDGFRAFLT3HRH3HRH4
SCHEMBL4819051 0.77 KDM4E (0.56) PDGFRBPDGFRAKDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7368572-B2 Acetylene derivatives as inhibitors of histone deacetylase PHARMACYCLICS, INC. (US) 2008-05-06 US disclosed