SCHEMBL14181069

SCHEMBL14181069

O=c1n(Cc2ccc(C(F)(F)F)cn2)nc2c(-c3ccc(Cl)cc3)c(-c3cccnc3)cnn12

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 10/20 0.57
PSD A5PKW4 3/20 0.38
CYP3A4 P08684 3/20 0.38
CYP2C9 P11712 3/20 0.36
CYP2C19 P33261 3/20 0.36
AVPR2 P30518 2/20 0.36
AVPR1A P37288 2/20 0.36
GRM2 Q14416 1/20 0.35
BRAF P15056 1/20 0.35
GPR119 Q8TDV5 1/20 0.34
CYP19A1 P11511 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4805900 0.91 CNR1 (0.62) CNR1CYP3A4CYP2C9CYP2C19AVPR2
SCHEMBL4807441 0.91 CNR1 (0.70) CNR1PSDCYP3A4CYP2C9CYP2C19
SCHEMBL14181067 0.91 CNR1 (0.70) CNR1PSDCYP3A4CYP2C9CYP2C19
SCHEMBL14181074 0.90 CNR1 (0.68) CNR1PSDCYP3A4CYP2C9CYP2C19
SCHEMBL14181126 0.86 CNR1 (0.68) CNR1PSDCYP3A4CYP2C9CYP2C19
SCHEMBL14181073 0.80 CNR1 (0.81) CNR1CYP3A4CYP2C9CYP2C19
SCHEMBL14180990 0.80 CNR1 (0.81) CNR1CYP3A4CYP2C9CYP2C19
SCHEMBL14181128 0.80 CNR1 (0.70) CNR1CYP3A4CYP2C9CYP2C19GPR119
SCHEMBL14181050 0.80 CNR1 (0.70) CNR1CYP3A4CYP2C9CYP2C19GPR119
SCHEMBL13114674 0.80 CNR1 (0.50) CNR1CYP3A4CYP2C9CYP2C19AVPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7378418-B2 Azabicyclic heterocycles as cannabinoid receptor modulators BRISTOL-MYERS SQUIBB COMPANY (US) 2008-05-27 US disclosed
US-7378418-B2 Azabicyclic heterocycles as cannabinoid receptor modulators BRISTOL-MYERS SQUIBB COMPANY (US) 2008-05-27 US disclosed