SCHEMBL14189656

SCHEMBL14189656

COC(=O)C(C)Cn1ccc2cc(-c3noc(-c4ccc(OC(C)C)c(Cl)c4)n3)ccc21

nearest known ligand 0.73

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 17/20 0.73
MAP4K4 O95819 3/20 0.52
MINK1 Q8N4C8 3/20 0.52
S1PR3 Q99500 4/20 0.51
DYRK3 O43781 1/20 0.51
MARK3 P27448 1/20 0.51
PLK1 P53350 1/20 0.51
MAP4K5 Q9Y4K4 1/20 0.51
PRKCD Q05655 1/20 0.49
S1PR5 Q9H228 1/20 0.48
CYP2C9 P11712 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1843851 1.00 S1PR1 (0.73) S1PR1MAP4K4MINK1S1PR3DYRK3
SCHEMBL1841883 0.92 S1PR1 (0.72) S1PR1MAP4K4MINK1S1PR3DYRK3
SCHEMBL400101 0.91 S1PR1 (0.78) S1PR1MAP4K4MINK1S1PR3DYRK3
SCHEMBL403510 0.91 S1PR1 (0.78) S1PR1MAP4K4MINK1S1PR3DYRK3
SCHEMBL10130558 0.85 S1PR1 (0.75) S1PR1MAP4K4MINK1S1PR3PRKCD
SCHEMBL398987 0.84 S1PR1 (1.00) S1PR1MAP4K4MINK1S1PR3S1PR5
SCHEMBL403328 0.84 S1PR1 (0.78) S1PR1MAP4K4MINK1S1PR3DYRK3
SCHEMBL401604 0.84 S1PR1 (0.92) S1PR1MAP4K4MINK1S1PR3S1PR5
SCHEMBL404571 0.83 S1PR1 (0.81) S1PR1MAP4K4MINK1S1PR3PRKCD
SCHEMBL403591 0.83 S1PR1 (0.90) S1PR1MAP4K4MINK1S1PR3S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008074821-A1 INDOLE DERIVATIVES AS S1P1 RECEPTOR AGONISTS GLAXO GROUP LIMITED (GB) 2008-06-26 WO disclosed