SCHEMBL14206751

SCHEMBL14206751

CCn1c([C@@H](C)NS(=O)(=O)c2ccc(Cl)cc2)nc2cc(Br)c(C(C)(F)F)cc21

nearest known ligand 0.68

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 20/20 0.68
CYP2D6 P10635 1/20 0.59
CYP2C19 P33261 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3449368 0.94 S1PR1 (0.72) S1PR1CYP2D6CYP2C19
SCHEMBL3451470 0.84 S1PR1 (0.77) S1PR1CYP2D6CYP2C19
SCHEMBL3449459 0.83 S1PR1 (0.88) S1PR1CYP2D6CYP2C19
SCHEMBL3449910 0.82 S1PR1 (0.84) S1PR1CYP2D6CYP2C19
SCHEMBL3449907 0.82 S1PR1 (0.84) S1PR1CYP2D6CYP2C19
SCHEMBL3450067 0.82 S1PR1 (0.75) S1PR1CYP2D6CYP2C19
SCHEMBL3449688 0.81 S1PR1 (0.76) S1PR1CYP2D6CYP2C19
SCHEMBL3450493 0.81 S1PR1 (0.86) S1PR1CYP2D6CYP2C19
SCHEMBL3449381 0.81 S1PR1 (0.85) S1PR1CYP2D6CYP2C19
SCHEMBL3450719 0.81 S1PR1 (1.00) S1PR1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008056150-A1 HETEROCYCLYC SULFONAMIDES HAVING EDG-I ANTAGONISTIC ACTIVITY ASTRAZENECA AB (SE) 2008-05-15 WO disclosed