SCHEMBL1421136

SCHEMBL1421136

CC(C)(C)OC(=O)NC1=N[C@H](C(C)(C)O)C[C@@](C)(c2ccc(F)c(-c3cncnc3)c2)S1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 3/20 0.36
BACE1 P56817 11/20 0.36
CTSD P07339 7/20 0.34
BACE2 Q9Y5Z0 7/20 0.34
CYP17A1 P05093 1/20 0.34
ACVR1B P36896 1/20 0.33
TGFBR1 P36897 1/20 0.33
ACVRL1 P37023 1/20 0.33
REN P00797 1/20 0.33
BRAF P15056 1/20 0.32
RORC P51449 1/20 0.32
EGLN2 Q96KS0 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1424309 1.00 ABL1 (0.36) ABL1BACE1CTSDBACE2CYP17A1
SCHEMBL1420673 0.91 BACE1 (0.39) ABL1BACE1CTSDBACE2CYP17A1
SCHEMBL4309373 0.89 ABL1 (0.36) ABL1BACE1CTSDBACE2REN
SCHEMBL1421083 0.86 SYK (0.37) ABL1BACE1CTSDBACE2CYP17A1
SCHEMBL1420814 0.84 BACE1 (0.35) BACE1CYP17A1BRAFRORC
SCHEMBL7990965 0.83 ABL1 (0.35) ABL1BACE1CTSDBACE2CYP17A1
SCHEMBL1421086 0.80 BACE1 (0.46) BACE1CTSDBACE2REN
SCHEMBL4313717 0.78 BACE1 (0.36) ABL1BACE1CTSDBACE2REN
SCHEMBL17004575 0.78 BACE1 (0.42) ABL1BACE1CTSDBACE2CYP17A1
SCHEMBL17004577 0.78 BACE1 (0.42) ABL1BACE1CTSDBACE2CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2297120-A1 AMINODIHYDROTHIAZINE DERIVATIVES AS BACE INHIBITORS FOR THE TREATMENT OF ALZHEIMER'S DISEASE Eli Lilly & Company (US) 2011-03-23 EP disclosed