SCHEMBL14212552

SCHEMBL14212552

Cc1onc(-c2ccccc2Cl)c1N(C)C=O

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 16/20 0.53
PTGS1 P23219 1/20 0.52
PTGS2 P35354 1/20 0.52
HSD17B10 Q99714 1/20 0.52
CYP3A4 P08684 2/20 0.50
CYP2C19 P33261 2/20 0.50
KMT2A Q03164 1/20 0.48
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
HTT P42858 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21119517 0.85 HSD17B10 (0.54) GPBAR1PTGS1PTGS2HSD17B10CYP3A4
SCHEMBL3724318 0.77 PTGS1 (0.57) GPBAR1PTGS1PTGS2HSD17B10CYP3A4
SCHEMBL10394013 0.74 PTGS1 (0.66) GPBAR1PTGS1PTGS2HSD17B10CYP3A4
SCHEMBL10083918 0.74 PTGS1 (0.66) GPBAR1PTGS1PTGS2HSD17B10CYP3A4
SCHEMBL27311110 0.73 PTGS1 (0.54) GPBAR1PTGS1PTGS2HSD17B10CYP2C19
SCHEMBL6254381 0.73 PTGS1 (0.47) GPBAR1PTGS1PTGS2HSD17B10CYP2C19
SCHEMBL21120027 0.73 HSD17B10 (0.56) GPBAR1PTGS1PTGS2HSD17B10CYP3A4
SCHEMBL10520547 0.72 HSD17B10 (0.76) GPBAR1HSD17B10CYP3A4CYP2C19KMT2A
SCHEMBL3545014 0.72 GPBAR1 (0.79) GPBAR1HSD17B10CYP3A4CYP2C19ALDH1A1
SCHEMBL14258658 0.71 PTGS1 (0.62) GPBAR1PTGS1PTGS2HSD17B10CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7378428-B2 Nitrogen-containing bicyclic compounds and drugs containing the same as the active ingredient ONO PHARMACEUTICAL CO., LTD. (JP) 2008-05-27 US disclosed