SCHEMBL14215741

SCHEMBL14215741

O=C(O)c1cc2ccc(-c3ccc(OCC4C(c5c(Cl)cccc5Cl)=NOC4C4CC4)cc3)cc2cn1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 16/20 0.51
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
ABL1 P00519 3/20 0.40
HSD17B13 Q7Z5P4 1/20 0.39
JAK2 O60674 1/20 0.38
TYK2 P29597 1/20 0.38
FABP1 P07148 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14215696 0.91 NR1H4 (0.44) NR1H4CYP1A2CYP2C9ABL1JAK2
SCHEMBL14215796 0.91 NR1H4 (0.43) NR1H4CYP1A2CYP2C9ABL1HSD17B13
SCHEMBL14215909 0.89 NR1H4 (0.52) NR1H4CYP1A2CYP2C9HSD17B13
SCHEMBL14215896 0.86 NR1H4 (0.51) NR1H4CYP1A2CYP2C9HSD17B13
SCHEMBL14215800 0.86 NR1H4 (0.51) NR1H4CYP1A2CYP2C9HSD17B13
SCHEMBL14215880 0.86 NR1H4 (0.58) NR1H4CYP1A2CYP2C9
SCHEMBL14215805 0.84 NR1H4 (0.45) NR1H4CYP1A2CYP2C9
SCHEMBL23474104 0.83 NR1H4 (0.36) NR1H4ABL1
SCHEMBL14215881 0.82 NR1H4 (0.37) NR1H4ABL1
SCHEMBL14215695 0.82 NR1H4 (0.45) NR1H4CYP1A2CYP2C9ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008051942-A2 FARNESOID X RECEPTOR AGONISTS SMITHKLINE BEECHAM CORPORATION (US) 2008-05-02 WO disclosed