SCHEMBL14224076

SCHEMBL14224076

c1ccc(Oc2cccc(-c3ncc(-c4ccnc(Nc5cccc(OCCCN6CCOCC6)c5)n4)[nH]3)c2)cc1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 4/20 0.49
BCR P11274 3/20 0.49
EPHX2 P34913 3/20 0.46
AIMP2 Q13155 2/20 0.46
ABL2 P42684 1/20 0.46
EGFR P00533 3/20 0.46
ITK Q08881 1/20 0.46
SYK P43405 4/20 0.45
SRC P12931 2/20 0.44
MTOR P42345 1/20 0.44
SMG1 Q96Q15 1/20 0.44
PRKCA P17252 1/20 0.44
PRKCD Q05655 1/20 0.44
RAF1 P04049 1/20 0.44
MAP2K1 Q02750 1/20 0.44
HDAC1 Q13547 1/20 0.42
MKNK1 Q9BUB5 1/20 0.42
BTK Q06187 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14224133 0.94 ABL1 (0.50) ABL1BCREPHX2AIMP2ABL2
SCHEMBL14224075 0.93 AIMP2 (0.48) ABL1BCRAIMP2EGFRSYK
SCHEMBL14195979 0.92 MTOR (0.54) ABL1BCREPHX2AIMP2ABL2
SCHEMBL14224454 0.92 AIMP2 (0.47) ABL1BCREPHX2AIMP2EGFR
SCHEMBL14224359 0.91 AIMP2 (0.48) ABL1BCRAIMP2EGFRSYK
SCHEMBL14224455 0.91 SYK (0.47) ABL1BCREPHX2AIMP2EGFR
SCHEMBL14224140 0.91 AIMP2 (0.50) ABL1BCRAIMP2EGFRSYK
SCHEMBL14196020 0.90 ABL1 (0.59) ABL1BCREPHX2AIMP2ABL2
SCHEMBL14224273 0.90 AIMP2 (0.45) ABL1BCRAIMP2EGFRSYK
SCHEMBL14224357 0.88 AIMP2 (0.48) ABL1BCRAIMP2EGFRSYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7361665-B2 Inhibitors of c-Jun N-terminal kinases (JNK) and other protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-04-22 US disclosed